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| Drug Name | NKT2152 |
| Trade Name | |
| Synonyms | NKT-2152|NKT 2152 |
| Drug Descriptions |
NKT2152 binds to HIF2A and blocks DNA binding, potentially resulting in decreased target gene expression, reduced tumor cell proliferation and tumor growth inhibiton (Cancer Res 2022;82(12_Suppl):Abstract nr 6330). |
| DrugClasses | HIF2A Inhibitor 6 |
| CAS Registry Number | NA |
| NCIT ID | C185419 |
| Therapy Name | Drugs | Efficacy Evidence | Clinical Trials |
|---|---|---|---|
| NKT2152 | NKT2152 | 0 | 1 |
| NKT2152 + Palbociclib | NKT2152 Palbociclib | 0 | 1 |
| NKT2152 + Palbociclib + PF-06801591 | NKT2152 PF-06801591 Palbociclib | 0 | 1 |