LOXO-435
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| Drug Name | LOXO-435 |
| Trade Name | |
| Synonyms | LOXO 435|LOXO435|LY3866288|LY 3866288|LY-3866288|Vepugratinib |
| Drug Descriptions |
LOXO-435 is an isoform-selective inhibitor of FGFR3 with potential antitumor activity (Cancer Res (2023) 83 (8_Supplement): CT119). |
| DrugClasses | FGFR3 Inhibitor 21 |
| CAS Registry Number | NA |
| NCIT ID | C192227 |
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| Therapy Name | Drugs | Efficacy Evidence | Clinical Trials |
|---|---|---|---|
| Enfortumab vedotin-ejfv + LOXO-435 + Pembrolizumab | Enfortumab vedotin-ejfv LOXO-435 Pembrolizumab | 0 | 1 |
| LOXO-435 | LOXO-435 | 0 | 1 |
| LOXO-435 + Pembrolizumab | LOXO-435 Pembrolizumab | 0 | 1 |
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