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| Drug Name | RMC-5127 |
| Trade Name | |
| Synonyms | RMC5127|RMC 5127 |
| Drug Descriptions |
RMC-5127 is a mutant-selective tri-complex inhibitor of RAS G12V, which potentially decreases tumor growth (Cancer Res (2024) 84 (6_Supplement): 3340). |
| DrugClasses | KRAS Inhibitor 31 |
| CAS Registry Number | NA |
| NCIT ID | NA |
| Therapy Name | Drugs | Efficacy Evidence | Clinical Trials |
|---|---|---|---|
| Cetuximab + RMC-5127 | Cetuximab RMC-5127 | 0 | 1 |
| Daraxonrasib + RMC-5127 | Daraxonrasib RMC-5127 | 0 | 1 |
| RMC-5127 | RMC-5127 | 0 | 1 |