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| Drug Name | Pelitinib |
| Trade Name | |
| Synonyms | EKB-569|WAY-EKB 569 |
| Drug Descriptions |
Pelitinib (EKB-569) is a nonselective inhibitor of EGFR, ERBB2 (HER2), and ERBB4 (HER4), which induces apoptosis and inhibits cell proliferation (PMID: 25988710). |
| DrugClasses | EGFR Inhibitor (Pan) 63 HER2 Inhibitor 44 |
| CAS Registry Number | 257933-82-7 |
| NCIT ID | C2713 |
| Therapy Name | Drugs | Efficacy Evidence | Clinical Trials |
|---|---|---|---|
| Futibatinib + Pelitinib | Futibatinib Pelitinib | 0 | 0 |
| Infigratinib + Pelitinib | Infigratinib Pelitinib | 0 | 0 |
| Pelitinib | Pelitinib | 0 | 0 |