Missing content? – Request curation!
Request curation for specific Genes, Variants, or PubMed publications.
Have questions, comments, or suggestions? - Let us know!
Email us at : ckbsupport@genomenon.com
| Drug Name | Tandutinib |
| Trade Name | |
| Synonyms | MLN518|CT53518|CT-53518|MLN-518 |
| Drug Descriptions |
Tandutinib (CT53518) is a tyrosine kinase inhibitor of FLT3, KIT, and PDGFRbeta, which inhibits cell proliferation and induces apoptosis (PMID: 12166950, PMID: 12124172, PMID: 27663390). |
| DrugClasses | FLT3 Inhibitor 69 KIT Inhibitor 57 PDGFR-beta Inhibitor 14 |
| CAS Registry Number | 387867-13-2 |
| NCIT ID | C48404 |
| Therapy Name | Drugs | Efficacy Evidence | Clinical Trials |
|---|---|---|---|
| Palbociclib + Tandutinib | Palbociclib Tandutinib | 1 | 0 |
| Tandutinib | Tandutinib | 8 | 0 |