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| Drug Name | Savolitinib |
| Trade Name | |
| Synonyms | HMPL-504|AZD6094|AZD-6094|Volitinib |
| Drug Descriptions |
Savolitinib (AZD6094) is a selective MET inhibitor, which inhibits MET kinase activity, resulting in decreased downstream signaling, and may inhibit growth of MET-expressing tumors (PMID: 25248999, PMID: 32027846, PMID: 30952639). |
| DrugClasses | MET Inhibitor 59 |
| CAS Registry Number | 1313725-88-0 |
| NCIT ID | C104732 |
| Therapy Name | Drugs | Efficacy Evidence | Clinical Trials |
|---|---|---|---|
| Afatinib + Savolitinib | Afatinib Savolitinib | 0 | 0 |
| Cetuximab + Savolitinib | Cetuximab Savolitinib | 0 | 1 |
| Durvalumab + Savolitinib | Durvalumab Savolitinib | 0 | 1 |
| Furmonertinib + Savolitinib | Furmonertinib Savolitinib | 0 | 0 |
| Gefitinib + Savolitinib | Gefitinib Savolitinib | 0 | 0 |
| Itraconazole + Savolitinib | Itraconazole Savolitinib | 0 | 0 |
| Lorlatinib + Savolitinib | Lorlatinib Savolitinib | 0 | 0 |
| Moxifloxacin + Savolitinib | Moxifloxacin Savolitinib | 0 | 0 |
| Osimertinib + Savolitinib | Osimertinib Savolitinib | 0 | 5 |
| Savolitinib | Savolitinib | 0 | 7 |