Pimitespib
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| Drug Name | Pimitespib |
| Trade Name | |
| Synonyms | TAS-116|TAS116 |
| Drug Descriptions |
Pimitespib (TAS-116) is a selective inhibitor of HSP90-alpha and HSP90-beta, which may lead to decreased tumor growth (PMID: 25416789, PMID: 31857719, PMID: 31536852, PMID: 30679388). |
| DrugClasses | HSP90 Inhibitor 35 |
| CAS Registry Number | 1260533-36-5 |
| NCIT ID | C134448 |
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| Therapy Name | Drugs | Efficacy Evidence | Clinical Trials |
|---|---|---|---|
| Imatinib + Pimitespib | Imatinib Pimitespib | 0 | 1 |
| Palbociclib + Pimitespib | Palbociclib Pimitespib | 0 | 1 |
| Pimitespib | Pimitespib | 0 | 2 |
| Pimitespib + Radiotherapy | Pimitespib Radiotherapy | 0 | 0 |
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