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| Drug Name | Tirapazamine |
| Trade Name | Tirazone |
| Synonyms | SR4233|WIN 59075 |
| Drug Descriptions |
Tirazone (tirapazamine) is a hypoxia-activated prodrug that induces DNA damage within hypoxic regions of tumors, potentially providing antineoplastic activity (PMID: 18666379, PMID: 32543771). |
| DrugClasses | |
| CAS Registry Number | 27314-97-2 |
| NCIT ID | C1464 |
| Therapy Name | Drugs | Efficacy Evidence | Clinical Trials |
|---|---|---|---|
| Pembrolizumab + Tirapazamine | Pembrolizumab Tirapazamine | 0 | 1 |
| Tirapazamine | Tirapazamine | 0 | 2 |