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Drug Name | INCB053914 |
Trade Name | |
Synonyms | INCB53914 |
Drug Descriptions |
INCB053914 is an ATP-competitive small molecule inhibitor of PIM kinases 1, 2, and 3, which may inhibit cell proliferation by blocking the phosphorylation of downstream targets (PMID: 29927999, PMID: 31725895). |
DrugClasses | PIM Inhibitor (Pan) 10 |
CAS Registry Number | 2088852-47-3 |
NCIT ID | C124226 |