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| Drug Name | MI-503 |
| Trade Name | |
| Synonyms | MI 503|MI503 |
| Drug Descriptions |
MI-503 inhibits the interaction between Menin and MLL (KMT2A), potentially decreasing growth and migration of tumor cells (PMID: 25817203, PMID: 29142068). |
| DrugClasses | MEN1-KMT2A Inhibitor 8 |
| CAS Registry Number | 1857417-13-0 |
| NCIT ID | NA |
| Therapy Name | Drugs | Efficacy Evidence | Clinical Trials |
|---|---|---|---|
| Enzalutamide + MI-503 | Enzalutamide MI-503 | 0 | 0 |
| Gilteritinib + MI-503 | Gilteritinib MI-503 | 0 | 0 |
| MI-503 | MI-503 | 1 | 0 |
| MI-503 + Ponatinib | MI-503 Ponatinib | 0 | 0 |
| MI-503 + Quizartinib | MI-503 Quizartinib | 0 | 0 |
| MI-503 + Sorafenib | MI-503 Sorafenib | 0 | 0 |