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| Drug Name | Amcenestrant |
| Trade Name | |
| Synonyms | SAR-439859|SAR 439859|SAR439859 |
| Drug Descriptions |
Amcenestrant (SAR439859) is a selective estrogen receptor degrader that down-regulates ER expression and signaling, resulting in tumor cell growth inhibition (Cancer Res 2017;77(4 Suppl):Abstract nr P3-04-05, PMID: 31721572). |
| DrugClasses | Hormone - Anti-estrogens 31 |
| CAS Registry Number | 2114339-57-8 |
| NCIT ID | C140354 |
| Therapy Name | Drugs | Efficacy Evidence | Clinical Trials |
|---|---|---|---|
| Abemaciclib + Amcenestrant | Abemaciclib Amcenestrant | 0 | 1 |
| Alpelisib + Amcenestrant | Alpelisib Amcenestrant | 0 | 1 |
| Amcenestrant | Amcenestrant | 0 | 5 |
| Amcenestrant + Everolimus | Amcenestrant Everolimus | 0 | 1 |
| Amcenestrant + Goserelin + Palbociclib | Amcenestrant Goserelin Palbociclib | 0 | 1 |
| Amcenestrant + Letrozole | Amcenestrant Letrozole | 0 | 1 |
| Amcenestrant + Midazolam | Amcenestrant Midazolam | 0 | 0 |
| Amcenestrant + Palbociclib | Amcenestrant Palbociclib | 0 | 2 |