Missing content? – Request curation!
Request curation for specific Genes, Variants, or PubMed publications.
Have questions, comments, or suggestions? - Let us know!
Email us at : ckbsupport@genomenon.com
Drug Name | ARV-771 |
Trade Name | |
Synonyms | ARV 771|ARV771 |
Drug Descriptions |
ARV-771 is a bifunctional molecule that targets BET proteins for proteolytic degradation, resulting in reduced target gene expression and potentially leading to increased apoptosis and reduced tumor growth (PMID: 31217338, PMID: 27274052, PMID: 30575820). |
DrugClasses | BET Inhibitor (Pan) 32 |
CAS Registry Number | 1949837-12-0 |
NCIT ID | NA |
Therapy Name | Drugs | Efficacy Evidence | Clinical Trials |
---|---|---|---|
ARV-771 | ARV-771 | 7 | 0 |
ARV-771 + Enzastaurin | ARV-771 Enzastaurin | 0 | 0 |