ARV-771
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| Drug Name | ARV-771 |
| Trade Name | |
| Synonyms | ARV 771|ARV771 |
| Drug Descriptions |
ARV-771 is a bifunctional molecule that targets BET proteins for proteolytic degradation, resulting in reduced target gene expression and potentially leading to increased apoptosis and reduced tumor growth (PMID: 31217338, PMID: 27274052, PMID: 30575820). |
| DrugClasses | BET Inhibitor (Pan) 33 |
| CAS Registry Number | 1949837-12-0 |
| NCIT ID | NA |
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| Therapy Name | Drugs | Efficacy Evidence | Clinical Trials |
|---|---|---|---|
| ARV-771 | ARV-771 | 7 | 0 |
| ARV-771 + Enzastaurin | ARV-771 Enzastaurin | 0 | 0 |
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