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Drug Name Triapine
Trade Name
Synonyms 3-AP|3-Apct|OCX-191|OCX 191|OCX191
Drug Descriptions

Triapine is an inhibitor of ribonucleotide reductase that blocks DNA synthesis, which potentially reduces cell viability and inhibits tumor growth (PMID: 10692563).

DrugClasses
CAS Registry Number 236392-56-6
NCIT ID C2242

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Therapy Name Drugs Efficacy Evidence Clinical Trials
Cediranib + Olaparib + Triapine Cediranib Olaparib Triapine 0 0
Cediranib + Triapine Cediranib Triapine 0 0
Cisplatin + Triapine Cisplatin Triapine 0 2
lutetium Lu 177 dotatate + Triapine Triapine lutetium Lu 177 dotatate 0 2
Olaparib + Triapine Olaparib Triapine 0 0
Temozolomide + Triapine Temozolomide Triapine 0 1
Triapine Triapine 0 1


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