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Drug Name | Olutasidenib |
Trade Name | Rezlidhia |
Synonyms | FT-2102 |
Drug Descriptions |
Rezlidhia (olutasidenib) targets IDH1 R132 mutations, leading to decreased 2HG production and potentially promoting differentiation and decreasing proliferation of IDH R132-mutant cancer cells (PMID: 31971798). Rezlidhia (olutasidenib) is FDA approved for use in adult patients with relapsed or refractory acute myeloid leukemia with a susceptible IDH1 mutation (FDA.gov). |
DrugClasses | IDH1 Inhibitor 8 |
CAS Registry Number | 1887014-12-1 |
NCIT ID | C129687 |