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| Drug Name | Relugolix |
| Trade Name | |
| Synonyms | TAK-385|Relumina |
| Drug Descriptions |
Relugolix (TAK-385) is a gonadotropin-releasing hormone antagonist, which binds to the gonadotropin-releasing hormone receptor, thereby preventing the secretion and release of luteinizing hormone and follicle stimulating hormone and possibly resulting in anti-tumor activity (PMID: 32469183). |
| DrugClasses | |
| CAS Registry Number | 737789-87-6 |
| NCIT ID | C114498 |
| Therapy Name | Drugs | Efficacy Evidence | Clinical Trials |
|---|---|---|---|
| Abiraterone + Prednisone + Relugolix | Abiraterone Prednisone Relugolix | 0 | 1 |
| Abiraterone + Relugolix | Abiraterone Relugolix | 0 | 1 |
| Bicalutamide + Pembrolizumab + Relugolix | Bicalutamide Pembrolizumab Relugolix | 0 | 1 |
| Darolutamide + Relugolix | Darolutamide Relugolix | 0 | 4 |
| Docetaxel + Relugolix | Docetaxel Relugolix | 0 | 2 |
| Enzalutamide + Relugolix | Enzalutamide Relugolix | 0 | 3 |
| Estradiol + Norethindrone + Relugolix | Estradiol Norethindrone Relugolix | 0 | 0 |
| Itraconazole + Relugolix | Itraconazole Relugolix | 0 | 1 |
| Relugolix | Relugolix | 0 | 11 |
| Relugolix + Ritonavir | Relugolix Ritonavir | 0 | 1 |