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| Drug Name | TTI-101 |
| Trade Name | |
| Synonyms | TTI101|TTI 101|C188-9 |
| Drug Descriptions |
TTI-101 (C188-9) is a small molecule that binds to STAT3 and inhibits signaling, potentially resulting in tumor cell death (PMID: 27027445, PMID: 32475130). |
| DrugClasses | STAT3 Inhibitor 26 |
| CAS Registry Number | 432001-19-9 |
| NCIT ID | C151932 |
| Therapy Name | Drugs | Efficacy Evidence | Clinical Trials |
|---|---|---|---|
| Atezolizumab + Bevacizumab + TTI-101 | Atezolizumab Bevacizumab TTI-101 | 0 | 1 |
| Fulvestrant + TTI-101 | Fulvestrant TTI-101 | 0 | 1 |
| Palbociclib + TTI-101 | Palbociclib TTI-101 | 0 | 1 |
| Pembrolizumab + TTI-101 | Pembrolizumab TTI-101 | 0 | 1 |
| Ribociclib + TTI-101 | Ribociclib TTI-101 | 0 | 1 |
| TTI-101 | TTI-101 | 0 | 4 |