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| Drug Name | Tunlametinib |
| Trade Name | |
| Synonyms | HL-085|HL085|HL 085 |
| Drug Descriptions |
Tunlametinib (HL-085) is a MEK inhibitor that may inhibit proliferation of tumor cells (Cancer Res 2019;79(13 Suppl):Abstract nr 4753). |
| DrugClasses | MEK inhibitor (Pan) 27 |
| CAS Registry Number | 1801756-06-8 |
| NCIT ID | C173437 |
| Therapy Name | Drugs | Efficacy Evidence | Clinical Trials |
|---|---|---|---|
| Adagrasib + Tunlametinib | Adagrasib Tunlametinib | 0 | 0 |
| Docetaxel + Tunlametinib | Docetaxel Tunlametinib | 0 | 0 |
| OKI-005 + Tunlametinib | OKI-005 Tunlametinib | 0 | 0 |
| SHP099 + Tunlametinib | SHP099 Tunlametinib | 0 | 0 |
| Sotorasib + Tunlametinib | Sotorasib Tunlametinib | 0 | 0 |
| Tunlametinib | Tunlametinib | 12 | 2 |
| Tunlametinib + Vemurafenib | Tunlametinib Vemurafenib | 4 | 0 |