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| Drug Name | KU-57788 |
| Trade Name | |
| Synonyms | KU57788|KU 57788 |
| Drug Descriptions |
KU-57788 is an inhibitor of DNA-PK, potentially inducing tumor cell death (PMID: 32439931). |
| DrugClasses | DNA_PK Inhibitor 9 |
| CAS Registry Number | 503468-95-9 |
| NCIT ID | NA |
| Therapy Name | Drugs | Efficacy Evidence | Clinical Trials |
|---|---|---|---|
| ARQ 751 + KU-57788 | ARQ 751 KU-57788 | 1 | 0 |
| GSK690693 + KU-57788 | GSK690693 KU-57788 | 1 | 0 |
| Ipatasertib + KU-57788 | Ipatasertib KU-57788 | 1 | 0 |
| KU-57788 | KU-57788 | 0 | 0 |
| KU-57788 + Miransertib | KU-57788 Miransertib | 2 | 0 |
| KU-57788 + MK2206 | KU-57788 MK2206 | 1 | 0 |