Missing content? – Request curation!
Request curation for specific Genes, Variants, or PubMed publications.
Have questions, comments, or suggestions? - Let us know!
Email us at : ckbsupport@genomenon.com
| Drug Name | DFF332 |
| Trade Name | |
| Synonyms | DFF 332|DFF-332 |
| Drug Descriptions |
DFF332 inhibits HIF-2alpha and blocks its DNA binding, which may lead to downregulation of HIF-2alpha target genes involved in tumor cell growth and survival (NCI Drug Dictionary). |
| DrugClasses | HIF2A Inhibitor 6 |
| CAS Registry Number | NA |
| NCIT ID | C180826 |
| Therapy Name | Drugs | Efficacy Evidence | Clinical Trials |
|---|---|---|---|
| DFF332 | DFF332 | 0 | 1 |
| DFF332 + Everolimus | DFF332 Everolimus | 0 | 1 |
| DFF332 + Spartalizumab + Taminadenant | DFF332 Spartalizumab Taminadenant | 0 | 1 |