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| Drug Name | Tipifarnib |
| Trade Name | |
| Synonyms | Zarnestra|R115777 |
| Drug Descriptions |
Zarnestra (tipifarnib) is a farnesyltransferase inhibitor, which alters post-translational modification and activation of Ras proteins, and may result in decreased tumor cell proliferation and reduced tumor growth (PMID: 11196150, PMID: 25323927, PMID: 32557577). |
| DrugClasses | Farnesyltransferase Inhibitor 4 |
| CAS Registry Number | 192185-72-1 |
| NCIT ID | C1703 |
| Therapy Name | Drugs | Efficacy Evidence | Clinical Trials |
|---|---|---|---|
| Adagrasib + Tipifarnib | Adagrasib Tipifarnib | 0 | 0 |
| Alpelisib + Tipifarnib | Alpelisib Tipifarnib | 11 | 1 |
| AZD8186 + Tipifarnib | AZD8186 Tipifarnib | 0 | 0 |
| Naxitamab + Tipifarnib | Naxitamab Tipifarnib | 0 | 1 |
| Osimertinib + Tipifarnib | Osimertinib Tipifarnib | 0 | 1 |
| Pictilisib + Tipifarnib | Pictilisib Tipifarnib | 0 | 0 |
| Sapanisertib + Tipifarnib | Sapanisertib Tipifarnib | 1 | 0 |
| SCH772984 + Tipifarnib | SCH772984 Tipifarnib | 2 | 0 |
| Sotorasib + Tipifarnib | Sotorasib Tipifarnib | 0 | 0 |
| Tipifarnib | Tipifarnib | 25 | 9 |
| Tipifarnib + Trametinib | Tipifarnib Trametinib | 2 | 0 |
| Tipifarnib + Ulixertinib | Tipifarnib Ulixertinib | 2 | 0 |
| Tipifarnib + Uprosertib | Tipifarnib Uprosertib | 1 | 0 |