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| Drug Name | Ensartinib |
| Trade Name | Ensacove |
| Synonyms | X-396 |
| Drug Descriptions |
Ensacove (ensartinib) is a small molecule inhibitor of ALK, which inhibits downstream signaling and potentially leads to decreased growth of ALK-expressing tumors (PMID: 21613408, PMID: 31628085). Ensacove (ensartinib) is FDA-approved for use in adult patients with ALK-positive locally advanced or metastatic non-small cell lung cancer who have not previously received an ALK-inhibitor (FDA.gov). |
| DrugClasses | ALK Inhibitor 33 |
| CAS Registry Number | 1370651-20-9 |
| NCIT ID | C102754 |
| Therapy Name | Drugs | Efficacy Evidence | Clinical Trials |
|---|---|---|---|
| Bevacizumab + Carboplatin + Ensartinib + Pemetrexed Disodium | Bevacizumab Carboplatin Ensartinib Pemetrexed Disodium | 0 | 1 |
| Carboplatin + Ensartinib | Carboplatin Ensartinib | 0 | 1 |
| Cisplatin + Ensartinib | Cisplatin Ensartinib | 0 | 1 |
| Denosumab + Ensartinib | Denosumab Ensartinib | 0 | 0 |
| Durvalumab + Ensartinib | Durvalumab Ensartinib | 0 | 1 |
| Ensartinib | Ensartinib | 47 | 8 |
| Ensartinib + Fruquintinib | Ensartinib Fruquintinib | 0 | 0 |
| Ensartinib + Pralsetinib | Ensartinib Pralsetinib | 0 | 0 |
| Ensartinib + Sirolimus | Ensartinib Sirolimus | 1 | 0 |