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Drug Name | CPI-0610 |
Trade Name | |
Synonyms | CPI0610|pelabresib |
Drug Descriptions |
CPI-0610 is a small molecule that binds to BET bromodomains and inhibits interaction with acetylated histones, resulting in regulation of BET-dependent gene expression and anti-tumor effects (PMID: 26815195, PMID: 31729905). |
DrugClasses | BET Inhibitor (Pan) 32 |
CAS Registry Number | 1380087-89-7 |
NCIT ID | C111901 |