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| Drug Name | Entospletinib |
| Trade Name | |
| Synonyms | GS-9973|GS 9973|GS9973 |
| Drug Descriptions |
Entospletinib (GS-9973) is a selective spleen tyrosine kinase (Syk) inhibitor, which in turn inhibits B-cell receptor signaling, leading to suppression of cell migration and inhibition of survival (PMID: 24779514, PMID: 32156743). |
| DrugClasses | SYK Inhibitor 15 |
| CAS Registry Number | 1229208-44-9 |
| NCIT ID | C105402 |