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| Drug Name | Subasumstat |
| Trade Name | |
| Synonyms | TAK981|TAK 981|TAK-981 |
| Drug Descriptions |
Subasumstat (TAK-981) is a small molecule inhibitor of the SUMO-activating enzyme (SAE), which may lead to activation of anti-tumor immune response and inhibition of tumor growth (PMID: 37420267). |
| DrugClasses | |
| CAS Registry Number | 1858276-04-6 |
| NCIT ID | C156270 |
| Therapy Name | Drugs | Efficacy Evidence | Clinical Trials |
|---|---|---|---|
| Avelumab + Subasumstat | Avelumab Subasumstat | 0 | 1 |
| Cetuximab + Subasumstat | Cetuximab Subasumstat | 0 | 1 |
| Daratumumab and hyaluronidase-fihj + Subasumstat | Daratumumab and hyaluronidase-fihj Subasumstat | 0 | 1 |
| Mezagitamab + Subasumstat | Mezagitamab Subasumstat | 0 | 1 |
| Pembrolizumab + Subasumstat | Pembrolizumab Subasumstat | 0 | 1 |
| Rituximab + Subasumstat | Rituximab Subasumstat | 0 | 1 |
| Subasumstat | Subasumstat | 0 | 2 |
| Subasumstat + Trametinib | Subasumstat Trametinib | 0 | 0 |