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| Drug Name | Lifirafenib |
| Trade Name | |
| Synonyms | BGB-283 |
| Drug Descriptions |
Lifirafenib (BGB-283) is a dual RAF kinase and EGFR inhibitor, which may lead to decreased tumor cell proliferation and reduced growth of tumors with activation of BRAF and/or EGFR (PMID: 26208524, PMID: 32182156). |
| DrugClasses | BRAF Inhibitor 26 EGFR Inhibitor (Pan) 63 |
| CAS Registry Number | 1446090-79-4 |
| NCIT ID | C124995 |
| Therapy Name | Drugs | Efficacy Evidence | Clinical Trials |
|---|---|---|---|
| Cetuximab + Lifirafenib | Cetuximab Lifirafenib | 1 | 0 |
| Lifirafenib | Lifirafenib | 12 | 1 |
| Lifirafenib + Mirdametinib | Lifirafenib Mirdametinib | 3 | 1 |
| Lifirafenib + MK-8353 | Lifirafenib MK-8353 | 2 | 0 |
| Lifirafenib + Pimasertib | Lifirafenib Pimasertib | 1 | 0 |
| Lifirafenib + SCH772984 | Lifirafenib SCH772984 | 3 | 0 |
| Lifirafenib + Selumetinib | Lifirafenib Selumetinib | 0 | 0 |
| Lifirafenib + Trametinib | Lifirafenib Trametinib | 4 | 0 |
| Lifirafenib + Ulixertinib | Lifirafenib Ulixertinib | 2 | 0 |
| Lifirafenib + Vemurafenib | Lifirafenib Vemurafenib | 2 | 0 |