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| Drug Name | VX-803 |
| Trade Name | |
| Synonyms | M4344|VX80|gartisertib |
| Drug Descriptions |
VX-803 (M4344) is an inhibitor of ATR that is used in combination with radiation or chemotherapy (PMID: 30645202, PMID: 31836456). |
| DrugClasses | ATR Inhibitor 16 |
| CAS Registry Number | 1613191-99-3 |
| NCIT ID | C129693 |
| Therapy Name | Drugs | Efficacy Evidence | Clinical Trials |
|---|---|---|---|
| Camptothecin + VX-803 | Camptothecin VX-803 | 0 | 0 |
| Carboplatin + VX-803 | Carboplatin VX-803 | 0 | 1 |
| Cisplatin + VX-803 | Cisplatin VX-803 | 0 | 0 |
| Etoposide + VX-803 | Etoposide VX-803 | 0 | 0 |
| Exatecan mesylate + VX-803 | Exatecan mesylate VX-803 | 0 | 0 |
| Gemcitabine + VX-803 | Gemcitabine VX-803 | 0 | 0 |
| Indotecan + VX-803 | Indotecan VX-803 | 0 | 0 |
| Irinotecan + VX-803 | Irinotecan VX-803 | 0 | 0 |
| MTX-1000 + VX-803 | MTX-1000 VX-803 | 0 | 0 |
| Niraparib + VX-803 | Niraparib VX-803 | 0 | 2 |
| SN-38 + VX-803 | SN-38 VX-803 | 0 | 0 |
| Talazoparib + VX-803 | Talazoparib VX-803 | 0 | 0 |
| Topotecan + VX-803 | Topotecan VX-803 | 0 | 0 |
| VX-803 | VX-803 | 0 | 1 |