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| Drug Name | Taselisib |
| Trade Name | |
| Synonyms | RG7606|GDC-0032|RG-7604|RO5537381 |
| Drug Descriptions |
Taselisib (GDC-0032) is a beta isoform-sparing PI3K inhibitor, with greater activity against oncogenic mutants of PIK3CA (PMID: 23662903, PMID: 31439579). |
| DrugClasses | PIK3CA inhibitor 27 PIK3CD inhibitor 27 PIK3CG inhibitor 10 |
| CAS Registry Number | 1282512-48-4 |
| NCIT ID | C116876 |