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| Drug Name | Telaglenastat |
| Trade Name | |
| Synonyms | CB-839 |
| Drug Descriptions |
Telaglenastat (CB-839) binds to and inhibits glutaminase, preventing the conversion of glutamine to glutamate, which results in a decrease in cell proliferation (PMID: 31980651). |
| DrugClasses | Glutaminase Inhibitor 3 |
| CAS Registry Number | 1439399-58-2 |
| NCIT ID | C114381 |