Zoldonrasib
Drug Detail

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Drug Name Zoldonrasib
Trade Name
Synonyms RMC 9805|RMC9805|RMC-9805|RM036|RM-036|RM 036
Drug Descriptions

Zoldonrasib (RMC-9805) inhibits KRAS G12D, which potentially results in reduced downstream signaling and proliferation, induction of apoptosis, and decreased tumor growth (Cancer Res 2023;83(7_Suppl):Abstract nr 526).

DrugClasses KRAS G12D Inhibitor 26
CAS Registry Number 3034802-05-3
NCIT ID C201828

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Therapy Name Drugs Efficacy Evidence Clinical Trials
Carboplatin + Daraxonrasib + Pemetrexed Disodium + Zoldonrasib Carboplatin Daraxonrasib Pemetrexed Disodium Zoldonrasib 0 1
Cetuximab + Ivonescimab + Zoldonrasib Cetuximab Ivonescimab Zoldonrasib 0 1
Cisplatin + Daraxonrasib + Pemetrexed Disodium + Zoldonrasib Cisplatin Daraxonrasib Pemetrexed Disodium Zoldonrasib 0 1
Daraxonrasib + Pembrolizumab + Zoldonrasib Daraxonrasib Pembrolizumab Zoldonrasib 0 1
Fluorouracil + Irinotecan + Leucovorin + Oxaliplatin + Zoldonrasib Fluorouracil Irinotecan Leucovorin Oxaliplatin Zoldonrasib 0 1
Gemcitabine + Nab-paclitaxel + Zoldonrasib Gemcitabine Nab-paclitaxel Zoldonrasib 0 1
Ivonescimab + Zoldonrasib Ivonescimab Zoldonrasib 0 1
TNG462 + Zoldonrasib TNG462 Zoldonrasib 0 1
Zoldonrasib Zoldonrasib 0 2


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