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| Drug Name | Entinostat |
| Trade Name | |
| Synonyms | HDAC inhibitor SNDX-275|MS 275 |
| Drug Descriptions |
Entinostat (MS-275) inhibits HDAC activity, with selectivity towards HDAC1, 2, and 3, which results in increased histone acetylation, and potentially leads to decreased tumor cell proliferation and tumor growth (PMID: 19724929, PMID: 17383217, PMID: 32503469). |
| DrugClasses | HDAC Inhibitor 45 |
| CAS Registry Number | 209783-80-2 |
| NCIT ID | C1863 |