Regorafenib
Drug Detail
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| Drug Name | Regorafenib |
| Trade Name | Stivarga |
| Synonyms | BAY 73-4506 |
| Drug Descriptions |
Stivarga (regorafenib) is an inhibitor of several kinases including VEGFR, RET, KIT, PDGFR and RAF, thereby inhibiting tumor angiogenesis and tumor cell proliferation (PMID: 24756792). Stivarga (regorafenib) is FDA approved for colorectal cancer, hepatocellular carcinoma, and GIST (FDA.gov). |
| DrugClasses | BRAF Inhibitor 26 CRAF Inhibitor 12 KIT Inhibitor 57 PDGFR Inhibitor (Pan) 30 RET Inhibitor 53 VEGFR Inhibitor (Pan) 36 VEGFR2 Inhibitor 37 |
| CAS Registry Number | 755037-03-7 |
| NCIT ID | C78204 |
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