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| Drug Name | Umbralisib |
| Trade Name | Ukoniq |
| Synonyms | RP5264|TGR-1202 |
| Drug Descriptions |
Ukoniq (umbralisib) inhibits PIK3CD and Casein Kinase 1 epsilon (CK1e), which decreases Akt phosphorylation and potentially reduces tumor cell viability (PMID: 33617893, PMID: 32634240, PMID: 30709431). |
| DrugClasses | PIK3CD inhibitor 27 |
| CAS Registry Number | 1532533-67-7 |
| NCIT ID | C104413 |