Tazemetostat
Drug Detail

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Drug Name Tazemetostat
Trade Name Tazverik
Synonyms EPZ6438|E-7438|EPZ-6438
Drug Descriptions

Tazverik (tazemetostat) binds to and inhibits EZH2, resulting in decreased tri-methylation of H3K27, which potentially leads to inhibition of cell proliferation and tumor growth (PMID: 23620515).

DrugClasses EZH2 inhibitor 20
CAS Registry Number 1403254-99-8
NCIT ID C107506

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Therapy Name Drugs Efficacy Evidence Clinical Trials
Abiraterone + Prednisone + Tazemetostat Abiraterone Prednisone Tazemetostat 0 1
Acalabrutinib + Tazemetostat Acalabrutinib Tazemetostat 0 2
Adagrasib + Tazemetostat Adagrasib Tazemetostat 0 0
AZD1390 + Tazemetostat AZD1390 Tazemetostat 0 0
Barasertib + Tazemetostat Barasertib Tazemetostat 0 0
Belinostat + Tazemetostat Belinostat Tazemetostat 0 1
Bendamustine + Rituximab + Tazemetostat Bendamustine Rituximab Tazemetostat 0 1
Binimetinib + Tazemetostat Binimetinib Tazemetostat 0 0
CC-92480 + Dexamethasone + Tazemetostat CC-92480 Dexamethasone Tazemetostat 0 1
Cetuximab + Encorafenib + Tazemetostat Cetuximab Encorafenib Tazemetostat 1 0
CPX-351 + Palbociclib + Tazemetostat CPX-351 Palbociclib Tazemetostat 0 1
CPX-351 + Tazemetostat CPX-351 Tazemetostat 0 1
Cyclophosphamide + Doxorubicin + Prednisolone + Rituximab + Tazemetostat + Vincristine Sulfate Cyclophosphamide Doxorubicin Prednisolone Rituximab Tazemetostat Vincristine Sulfate 0 1
Cyclophosphamide + Doxorubicin + Prednisone + Tazemetostat + Vincristine Sulfate Cyclophosphamide Doxorubicin Prednisone Tazemetostat Vincristine Sulfate 0 1
Dabrafenib + Tazemetostat + Trametinib Dabrafenib Tazemetostat Trametinib 0 1
Daratumumab + Dexamethasone + Pomalidomide + Tazemetostat Daratumumab Dexamethasone Pomalidomide Tazemetostat 0 1
Daratumumab and hyaluronidase-fihj + Dexamethasone + Pomalidomide + Tazemetostat Daratumumab and hyaluronidase-fihj Dexamethasone Pomalidomide Tazemetostat 0 1
Dexamethasone + Tazemetostat Dexamethasone Tazemetostat 0 0
Doxorubicin + Tazemetostat Doxorubicin Tazemetostat 0 1
Durvalumab + Tazemetostat Durvalumab Tazemetostat 0 1
Encorafenib + Tazemetostat Encorafenib Tazemetostat 1 0
Enzalutamide + Tazemetostat Enzalutamide Tazemetostat 0 1
Epcoritamab-bysp + Tazemetostat Epcoritamab-bysp Tazemetostat 0 1
Everolimus + Tazemetostat Everolimus Tazemetostat 0 0
Fluconazole + Tazemetostat Fluconazole Tazemetostat 0 1
Ibrutinib + Tazemetostat Ibrutinib Tazemetostat 0 0
Idelalisib + Tazemetostat Idelalisib Tazemetostat 0 0
Ipilimumab + Nivolumab + Tazemetostat Ipilimumab Nivolumab Tazemetostat 0 1
Itraconazole + Tazemetostat Itraconazole Tazemetostat 0 1
LAM-003 + Tazemetostat LAM-003 Tazemetostat 1 0
Lenalidomide + Rituximab + Tazemetostat Lenalidomide Rituximab Tazemetostat 0 1
Lenalidomide + Tafasitamab-cxix + Tazemetostat Lenalidomide Tafasitamab-cxix Tazemetostat 0 2
Lenalidomide + Tazemetostat Lenalidomide Tazemetostat 0 1
MK2206 + Tazemetostat MK2206 Tazemetostat 0 0
Mosunetuzumab-axgb + Tazemetostat Mosunetuzumab-axgb Tazemetostat 0 2
MRTX-1133 + Tazemetostat MRTX-1133 Tazemetostat 0 0
Nilotinib + Tazemetostat Nilotinib Tazemetostat 0 0
Obinutuzumab + Rituximab + Tazemetostat + Zanubrutinib Obinutuzumab Rituximab Tazemetostat Zanubrutinib 0 1
Omeprazole + Repaglinide + Tazemetostat Omeprazole Repaglinide Tazemetostat 0 1
Panobinostat + Tazemetostat Panobinostat Tazemetostat 1 0
Pembrolizumab + Tazemetostat Pembrolizumab Tazemetostat 0 3
Pembrolizumab + Tazemetostat + Topotecan Pembrolizumab Tazemetostat Topotecan 0 1
Rifampin + Tazemetostat Rifampin Tazemetostat 0 1
Rituximab + Tazemetostat Rituximab Tazemetostat 0 1
Selumetinib + Tazemetostat Selumetinib Tazemetostat 0 0
Talazoparib + Tazemetostat Talazoparib Tazemetostat 0 1
Tamatinib + Tazemetostat Tamatinib Tazemetostat 0 0
Tazemetostat Tazemetostat 3 16
Tazemetostat + Trametinib Tazemetostat Trametinib 1 0
Tazemetostat + Ublituximab + Umbralisib Tazemetostat Ublituximab Umbralisib 0 1
Tazemetostat + Venetoclax Tazemetostat Venetoclax 0 1
Tazemetostat + zandelisib Tazemetostat zandelisib 0 1


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