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Drug Name Zanidatamab
Trade Name Ziihera
Synonyms ZW-25|ZW25|Zanidatamab-hrii
Drug Descriptions

Ziihera (zanidatamab) is a bispecific antibody targeting ERBB2 (HER2), which induces anti-tumor immune response against Erbb2 (Her2)-expressing tumors (Ann Oncol 2017, Vol 28, Suppl 5, Abstract # 255P, PMID: 32054397). Ziihera (zanidatamab) is FDA-approved for use in patients with unresectable or metastatic ERBB2 (HER2)-positive (IHC 3+) biliary tract cancer (FDA.gov).

DrugClasses HER2 (ERBB2) Antibody 76
CAS Registry Number 2169946-15-8
NCIT ID C130010

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Therapy Name Drugs Efficacy Evidence Clinical Trials
Bevacizumab + Fluorouracil + Leucovorin + Oxaliplatin + Zanidatamab Bevacizumab Fluorouracil Leucovorin Oxaliplatin Zanidatamab 0 1
Capecitabine + Cisplatin + Zanidatamab Capecitabine Cisplatin Zanidatamab 0 0
Capecitabine + Oxaliplatin + Tislelizumab + Zanidatamab Capecitabine Oxaliplatin Tislelizumab Zanidatamab 0 1
Capecitabine + Oxaliplatin + Zanidatamab Capecitabine Oxaliplatin Zanidatamab 0 2
Capecitabine + Zanidatamab Capecitabine Zanidatamab 0 2
Capmatinib + Zanidatamab Capmatinib Zanidatamab 0 0
Cisplatin + Durvalumab + Gemcitabine + Zanidatamab Cisplatin Durvalumab Gemcitabine Zanidatamab 0 1
Cisplatin + Fluorouracil + Leucovorin + Zanidatamab Cisplatin Fluorouracil Leucovorin Zanidatamab 0 0
Cisplatin + Fluorouracil + Tislelizumab + Zanidatamab Cisplatin Fluorouracil Tislelizumab Zanidatamab 0 1
Cisplatin + Fluorouracil + Zanidatamab Cisplatin Fluorouracil Zanidatamab 0 2
Cisplatin + Gemcitabine + Pembrolizumab + Zanidatamab Cisplatin Gemcitabine Pembrolizumab Zanidatamab 0 1
Cisplatin + Gemcitabine + Zanidatamab Cisplatin Gemcitabine Zanidatamab 0 1
Crizotinib + Zanidatamab Crizotinib Zanidatamab 0 0
Docetaxel + Zanidatamab Docetaxel Zanidatamab 0 0
Eribulin + Zanidatamab Eribulin Zanidatamab 0 1
Evorpacept + Zanidatamab Evorpacept Zanidatamab 0 1
Fluorouracil + Leucovorin + Oxaliplatin + Zanidatamab Fluorouracil Leucovorin Oxaliplatin Zanidatamab 0 1
Fulvestrant + Palbociclib + Zanidatamab Fulvestrant Palbociclib Zanidatamab 0 1
Gemcitabine + Zanidatamab Gemcitabine Zanidatamab 0 1
JQ1 + Zanidatamab JQ1 Zanidatamab 0 0
Letrozole + Tamoxifen + Zanidatamab Letrozole Tamoxifen Zanidatamab 0 0
Letrozole + Zanidatamab Letrozole Zanidatamab 0 1
Paclitaxel + Ramucirumab + Zanidatamab Paclitaxel Ramucirumab Zanidatamab 0 1
Paclitaxel + Zanidatamab Paclitaxel Zanidatamab 0 1
Tamoxifen + Zanidatamab Tamoxifen Zanidatamab 0 1
Vinorelbine + Zanidatamab Vinorelbine Zanidatamab 0 2
Zanidatamab Zanidatamab 0 7


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